Emapunil (AC5216)

Emapunil (AC5216)

【产品别名】AC 5216;XBD-173;

【CAS号】 226954-04-7

【目录编号】 3HC-8

【纯度】 >98%

【分子式】 C23H23N5O2

【分子量】 401.46


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Emapunil (AC5216) 详细介绍

Emapunil (AC-5216XBD-173) is an anxiolytic drug which acts as a selective agonist at the peripheral benzodiazepine receptor, also known as the mitochondrial 18 kDa translocator protein or TSPO. This protein has multiple functions, among which is regulation of steroidogenesis, particularly the production of neuroactive steroids such as allopregnanolone in the brain. In both animal and human trials, emapunil produced fast acting anxiolytic and anti-panic effects, without producing sedation or withdrawal symptoms following cessation of use.Emapunil is also used in its 11radiolabelled form to map the distribution of TSPO receptors in the brain.

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